LN-654714
4-DesMethyl Istradefylline , 0.97 , 160434-48-0
Update time: 2023-04-23
PRODUCT Properties
| Boiling point: | 604.8±65.0 °C(Predicted) |
| Density | 1.30±0.1 g/cm3(Predicted) |
| pka | 9.88±0.31(Predicted) |
Description and Uses
4-Desmethyl Istradefylline is an impurity of Istradefylline (I927000), a selective A(2A) antagonist used in the treatment of Parkinson’s disease. 4-Desmethyl Istradefylline have also been shown to exhibit inhibitory potency towards adenosine A2A receptors and is classified as its an adenosine A2A receptor antagonist.




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