M2403335
ERK5-IN-1 , 99% , 1435488-37-1
Synonym(s):
11-Cyclopentyl-2-((2-ethoxy-4-(4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl)-phenyl)amino)-5-methyl-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one;ERK5-IN-1
CAS NO.：1435488-37-1
Empirical Formula: C36H46N8O3
Molecular Weight: 638.8
MDL number:
EINECS: 604-604-1
| Pack Size | Price | Stock | Quantity |
| 5mg | RMB1482.40 | In Stock |
|
| others | Enquire |
Update time: 2022-07-08
PRODUCT Properties
| storage temp. | -20°C |
| solubility | ≥31.95 mg/mL in DMSO; insoluble in H2O; ≥86.6 mg/mL in EtOH |
| form | powder |
| color | white to beige |
| InChIKey | XVBGRTMNFNMINE-UHFFFAOYSA-N |
| SMILES | N7(CCN(CC7)C)C1CCN(CC1)C(=O)c2cc(c(cc2)Nc3nc4[n](c6c([c]([n](c4cn3)C)=O)cccc6)C5CCCC5)OCC |
Description and Uses
ERK5-IN-1 is a potent selective ERK5 inhibitor, inhibiting EGFR-induced ERK5 autophosphorylation and ERK5 enzymatic activity. Orally bioavailable.
Safety
| Symbol(GHS) |  GHS07 |
| Signal word | Warning |
| Hazard statements | H315-H319 |
| Precautionary statements | P305+P351+P338 |
| WGK Germany | WGK 3 |
| HS Code | 2933599590 |
| Storage Class | 11 - Combustible Solids |
| Hazard Classifications | Eye Irrit. 2 Skin Irrit. 2 |
