S9191814
solid,≥98%(HPLC) , 80880-90-6
Synonym(s):
4,9-Dihydro-3-methyl-4-[(4-methyl-1-piperazinyl)acetyl]-10H-thieno[3,4-b][1,5]benzodiazepin-10-one dihydrochloride
CAS NO.：80880-90-6
Empirical Formula: C19H22N4O2S
Molecular Weight: 370.475
MDL number: MFCD00083208
| Pack Size | Price | Stock | Quantity |
| 10mg | RMB686.50 | In Stock |
|
| 25mg | RMB1437.18 | In Stock |
|
| 100mg | RMB4357.14 | In Stock |
|
| others | Enquire |
Update time: 2022-07-08
PRODUCT Properties
| Melting point: | 263-264° |
| Boiling point: | 544.7±50.0 °C(Predicted) |
| Density | 1.281±0.06 g/cm3(Predicted) |
| solubility | H2O: >10 mg/mL |
| form | solid |
| pka | 12.48±0.20(Predicted) |
| color | white |
Description and Uses
Telenzepine is an antimuscarinic agent with Kis of 0.94 nM (M1 mAChR) and 17.8 nM (M2 mAChR) binding to muscarinic receptors. Telenzepine effectively blocks synaptic transmission promoted by muscarinic or M1 receptor agonists. Thus, Telenzepine can reduce the amplitude of extracellular slow excitatory postsynaptic potentials (EC50=38 nM) and slow inhibitory postsynaptic potentials (EC50=253 nM)[1].
Safety
| WGK Germany | 3 |
