≥97%(HPLC) , 150375-75-0

Synonym(s):
(2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide;SR49059

CAS NO.：150375-75-0

Empirical Formula: C28H27Cl2N3O7S

Molecular Weight: 620.5

MDL number: MFCD00922133

PRODUCT Properties

• Melting point: 158-160oC
• Boiling point: 868.0±75.0 °C(Predicted)
• Density: 1.499±0.06 g/cm3(Predicted)
• storage temp.: 2-8°C
• solubility: DMSO: ≥10mg/mL
• pka: 10.95±0.40(Predicted)
• form: powder
• color: white to off-white
• optical activity: [α]/D -180 to -190°, c = 0.3 in chloroform-d
• Stability: Hygroscopic

Description and Uses

Relcovaptan is a selective vasopressin-1a receptor antagonist that prevents cellular swelling and provides treatment for post-traumatic brain edema.

Safety

• Symbol(GHS): GHS07
• Signal word: Warning
• Hazard statements: H302-H317
• Precautionary statements: P280-P305+P351+P338
• WGK Germany: nwg